Tianeptine FA cas 72797-41-2
Product introduction:
Product name: Tianeptine FA
Chemical name: Einecs 276-851-9, TPI-1062, Tianeptin
Cas: 72797-41-2
Purity: 99.0%min
Appearance: White or almost white micro crystalline powder
MF: C23H29ClN2O4S
Molecular Weight: 436.95
Solubility: Insoluble in the water and methanol
Residue on ignation: Not more than 0.2%
Tianeptine Acid is a drug used primarily in the treatment of major depressive disorder, although it may also be used to treat asthma or irritable bowel syndrome. Chemically it is a tricyclic antidepressant (TCA), but it has different pharmacological properties than typical TCAs as recent research suggests that tianeptine produces its antidepressant effects through indirect alteration of glutamate receptor activity (i.e., AMPA receptors and NMDA receptors) and release of BDNF, in turn affecting neural plasticity.
Application: Tianeptine FA cas 72797-41-2 has antidepressant and anxiolytic (anti-anxiety) properties with a relative lack of sedative, anticholinergic and cardiovascular adverse effects, thus suggesting it is particularly suitable for use in the elderly and in those following alcohol withdrawal; such persons can be more sensitive to the adverse effects of psychotropic drugs. Recent results indicate possible anticonvulsant (anti-seizure) and analgesic (painkilling) activity of tieneptine via immediate or downstream modulation of adenosine A1 receptors (as the effects could be experimentally blocked by antagonists of this receptor).